EZM0414
Product Specifications
CAS Number
2411748-50-8
Target
Histone Methyltransferase
Related Pathways
Chromatin/Epigenetic
Purity
0.9958
Bioactivity
EZM0414 is a potent and selective, orally bioavailable inhibitor of SETD2 with an IC50 of 18 nM in biochemical assays and 34 nM in cellular assays, potentially useful for researching relapsed or refractory multiple myeloma and diffuse large B-cell lymphoma [1].
Smiles
[H][C@@]1(CCC[C@H](C1)NC(=O)c1cc2c(F)ccc(C)c2[nH]1)N1CCN(CC1)C(C)=O
Molecular Formula
C22H29FN4O2
Molecular Weight
400.49
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
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