Deulumateperone
Deulumateperone is a deuterium labeled Lumateperone (HY-17637) . Lumateperone is the orally active 5-HT2A receptor antagonist (Ki = 0.54 nM) and the modulator for dopamine receptor that exhibits antipsychotic and antineoplastic activities[1].
Product Specifications
CAS Number
[2102683-75-8]
UNSPSC
12352005
Target
5-HT Receptor; Dopamine Receptor; Isotope-Labeled Compounds
Related Pathways
GPCR/G Protein; Neuronal Signaling; Others
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Smiles
CN1C2=C3C([C@@]4([H])[C@@](CCN(C4)CCCC(C5=CC=C(C=C5)F)=O)([H])N3CC1([2H])[2H])=CC=C2
Molecular Formula
C24H26D2FN3O
Molecular Weight
395.51
References & Citations
[1]Oguma T, et al., Clinical Pipelines for Alzheimer's Disease Psychosis and Agitation. Chem Pharm Bull (Tokyo) . 2024;72 (7) :610-617.
Shipping Conditions
Room temperature
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-172425/
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
5-HT2 Receptor
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items