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TEAD-IN-9

Product Specifications

Target

YAP

Related Pathways

Stem Cells

Bioactivity

TEAD-IN-9 (compound 17) is a TEAD1 inhibitor with an IC50 of 0.29 μM. It targets the palmitoyl pocket of TEAD, effectively inhibiting the binding of YAP-TEAD and blocking the transcriptional function of YAP-TEAD.

Molecular Formula

C23H23F3N3O3P

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

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