RP-72540
RP-72540 is a selective cholecystokinin B receptor (CCKB) antagonist with high affinity for gastrin binding sites and a 200-fold selectivity over CCKA receptors. It inhibits [3H]pCCK-8 binding in vitro but exhibits minimal brain penetration in vivo, making it a useful tool for studying peripheral CCKB/gastrin receptor functions in gastrointestinal research.
Product Specifications
CAS Number
139088-45-2
Field of Research
Pharmacology & Drug Discovery
Smiles
N (CC (N (C) C1=CC=CC=C1) =O) (C (CNC (NC2=CC (C (C (O) =O) C) =CC=C2) =O) =O) C3=CC (OC) =CC=C3
Molecular Formula
C28H30N4O6
Molecular Weight
518.56
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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