APJ receptor agonist 1
Product Specifications
CAS Number
2287153-38-0
Target
Apelin receptor|||Others
Related Pathways
GPCR/G Protein|||Others
Bioactivity
APJ receptor agonist 1, a potent biphenyl acid derivative, acts as an agonist (EC50 of 0.093 nM and 0.12 nM for human and rat APJ receptors, respectively) for the APJ receptor (APJ-R) . It exhibits significant in vitro potency towards apelin-13, the endogenous peptidic ligand for the APJ receptor. APJ receptor agonist 1 holds promise for heart failure research.
Smiles
CCCC(NC(=O)c1ccc(c(c1)C(O)=O)-c1c(Cl)cccc1-c1nc2ccccc2[nH]1)c1ccccc1
Molecular Formula
C31H26ClN3O3
Molecular Weight
524.02
Shipping Conditions
Cool pack
Storage Temperature
-20°C
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