SER-601

SER-601 is a potent and selective peripheral cannabinoid (CB2) receptor agonist with a Ki of 6.3 nM. SER-601 has analgesic and antidiabetic properties and can be used for relevant research[1].

Product Specifications

CAS Number

[1048038-90-9]

UNSPSC

12352005

Target

Cannabinoid Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein; Neuronal Signaling

Field of Research

Neurological Disease

Assay Protocol

https://www.medchemexpress.com/ser-601.html

Smiles

O=C(C(C(C1=CC(C(C)C)=CC=C12)=O)=CN2CCCCC)NC3(C[C@@H](C4)C5)C[C@@H]5C[C@@H]4C3

Molecular Formula

C28H38N2O2

Molecular Weight

434.61

References & Citations

[1]Pasquini S, et al. Investigations on the 4-quinolone-3-carboxylic acid motif. 2. Synthesis and structure-activity relationship of potent and selective cannabinoid-2 receptor agonists endowed with analgesic activity in vivo. J Med Chem. 2008 Aug 28;51 (16) :5075-84.