A 987306
Product Specifications
CAS Number
1082954-71-9
Target
Histamine Receptor, Others
Related Pathways
GPCR/G Protein, Others, Immunology/Inflammation, Neuroscience
Bioactivity
A-987306 is a potent and orally bioavailable histamine H4 antagonist with Kis of 3.4 nM and 5.8 nM for rat H4 and human H4, respectively. A-987306 exhibits anti-inflammatory activity in a mouse peritonitis model [1].
Smiles
NC=1N=C2C=3[C@]4([C@@](OC3CCC2=C(N1)N5CCNCC5)(CCCC4)[H])[H]
Molecular Formula
C18H25N5O
Molecular Weight
327.42
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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