DKM 2-93
DKM 2-93 is a relatively selective inhibitor of UBA5 with an IC50 of 430 μM.
Product Specifications
CAS Number
[65836-72-8]
UNSPSC
12352005
Hazard Statement
H301, H311, H331, H341
Target
E1/E2/E3 Enzyme
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/DKM_2-93.html
Purity
98.76
Solubility
DMSO : 125 mg/mL (ultrasonic)
Smiles
O=C(NCC1=CC=C(OC)C(OC)=C1)CCl
Molecular Formula
C11H14ClNO3
Molecular Weight
243.69
Precautions
H301, H311, H331, H341
References & Citations
[1]Roberts AM, et al. Chemoproteomic Screening of Covalent Ligands Reveals UBA5 As a Novel Pancreatic Cancer Target. ACS Chem Biol. 2017 Apr 21;12 (4) :899-904.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Curated Selection
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