Endoxifen (hydrochloride)
Endoxifen hydrochloride is a key active metabolite of Tamoxifen (TAM) with higher affinity and specificity to estrogen receptor that also inhibits aromatase activity. Endoxifen hydrochloride has the potential for breast cancer study[1][2].
Product Specifications
CAS Number
1197194-41-4
UNSPSC
12352005
Target
Cytochrome P450; Drug Metabolite; Estrogen Receptor/ERR; Parasite
Type
Reference compound
Related Pathways
Anti-infection; Metabolic Enzyme/Protease; Vitamin D Related/Nuclear Receptor
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/Endoxifen-hydrochloride.html
Purity
98.04
Solubility
DMSO : ≥ 35 mg/mL|H2O : < 0.1 mg/mL
Smiles
OC1=CC=C(/C(C2=CC=C(OCCNC)C=C2)=C(C3=CC=CC=C3)\CC)C=C1.[H]Cl
Molecular Formula
C25H28ClNO2
Molecular Weight
409.95
References & Citations
Shipping Conditions
Room Temperature
Storage Conditions
4°C (Powder, sealed storage, away from moisture)
Scientific Category
Reference compound1
Clinical Information
Phase 3
Isoform
Aromatase/CYP19A1
Available Sizes
Frequently Asked Questions
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