Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

MELK-8a (hydrochloride)

MELK-8a hydrochloride is a novel maternal embryonic leucine zipper kinase (MELK) inhibitor with an IC50 of 2 nM.

Product Specifications

CAS Number

2096992-20-8

Product Name Alternative

NVS-MELK8a (hydrochloride)

UNSPSC

12352005

Target

MELK

Type

Reference compound

Related Pathways

PI3K/Akt/mTOR

Applications

Cancer-Kinase/protease

Field of Research

Cancer

Assay Protocol

https://www.medchemexpress.com/MELK-8a-hydrochloride.html

Purity

99.31

Solubility

DMSO : 8.6 mg/mL (ultrasonic; warming) |H2O : ≥ 100 mg/mL

Smiles

CN(CC1)CCN1C2=CC=C(N3C=C(C4=CC=NC=C4OCC5CCNCC5)C=N3)C=C2.Cl

Molecular Formula

C25H33ClN6O

Molecular Weight

469.02

References & Citations

[1]Touré BB, et al. Toward the Validation of Maternal Embryonic Leucine Zipper Kinase: Discovery, Optimization of Highly Potent and Selective Inhibitors, and Preliminary Biology Insight. J Med Chem. 2016 May 26;59 (10) :4711-23.

Shipping Conditions

Room Temperature

Storage Conditions

4°C (Powder, sealed storage, away from moisture)

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Available Sizes

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

Frozen Tissue Sections, Neurovascular bundle
CS631922 5x 5 µm

Frozen Tissue Sections, Neurovascular bundle

Sign In for Pricing
View Details
LLCFC1 (NM_178829) Human Over-expression Lysate
LY432125 100 µg

LLCFC1 (NM_178829) Human Over-expression Lysate

Sign In for Pricing
View Details
Bulk Anti-Human CD56 (ERIC-1) Antibody
ICH1015-100mg 100 mg

Bulk Anti-Human CD56 (ERIC-1) Antibody

Sign In for Pricing
View Details
Frozen Tissue Blocks, Colon
CB507806 1 Block

Frozen Tissue Blocks, Colon

Sign In for Pricing
View Details
PTPN20B (PTPN20) (NM_001042363) Human Over-expression Lysate
LY420852 100 µg

PTPN20B (PTPN20) (NM_001042363) Human Over-expression Lysate

Sign In for Pricing
View Details
Pet1 Recombinant Rabbit Monoclonal Antibody [PSH07-77]
HA722893 100 µL

Pet1 Recombinant Rabbit Monoclonal Antibody [PSH07-77]

Sign In for Pricing
View Details