(Rac) -PD0299685
(Rac) -PD0299685 is a Ca (2+) channel α2δ ligand that was investigated for relieving interstitial cystitis pain in a randomized, double-blind, placebo-controlled phase IIa study. (Rac) -PD0299685 demonstrated a clinically significant reduction in daily worst pain severity scores at the 60 mg dose compared to placebo. (Rac) -PD0299685 is also a potent voltage-dependent calcium channel inhibitor for the study of retina-related diseases.
Product Specifications
CAS Number
[313651-02-4]
UNSPSC
12352211
Target
Calcium Channel
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/rac-pd0299685.html
Smiles
O=C(CC(CC(CCC)C)CN)O
Molecular Formula
C10H21NO2
Molecular Weight
187.28
References & Citations
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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