BCRP-IN-1
BCRP-IN-1 (compound 48) is a potent inhibitor of breast cancer resistance protein (BCRP), with IC50s of 2.92 μM and 2.46 μM in Hoechst 33342 assay and Pheophorbide A assay, respectively[1].
Product Specifications
CAS Number
765899-28-3
UNSPSC
12352005
Hazard Statement
H302-H315-H319
Target
BCRP
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/bcrp-in-1-1.html
Smiles
O=[N+](C1=CC=C(NC2=C3C=C(OC)C(OC)=CC3=NC=N2)C=C1)[O-]
Molecular Formula
C16H14N4O4
Molecular Weight
326.31
Precautions
P264-P270-P280-P302+P352-P305+P351+P338-P330-P362+P364-P501
References & Citations
[1]"Kapil Juvale, et al. Investigation of quinazolines as inhibitors of breast cancer resistance protein (ABCG2) . Bioorg Med Chem. 2013 Dec 15;21 (24) :7858-73. "
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Frequently Asked Questions
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