Tazemetostat (EPZ-6438)
Product Specifications
CAS Number
1403254-99-8
Synonyms
E7438
Target
Histone Methyltransferase
Applications
Epigenetics
Smiles
CCN (C1CCOCC1) C2=CC (=CC (=C2C) C (=O) NCC3=C (C=C (NC3=O) C) C) C4=CC=C (C=C4) CN5CCOCC5
Molecular Formula
C34H44N4O4
Additionnal Information
Tazemetostat (EPZ-6438, E7438) is a potent, and selective EZH2 inhibitor with Ki and IC50 of 2.5 nM and 11 nM in cell-free assays, exhibiting a 35-fold selectivity versus EZH1 and >4,500-fold selectivity relative to 14 other HMTs.
Storage Conditions
2 years -80 in solvent
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