Ivarmacitinib
Product Specifications
CAS Number
1445987-21-2
Synonyms
SHR0302
Target
JAK
Applications
Angiogenesis
Molecular Formula
C18H22N8O2S
Additionnal Information
Ivarmacitinib (SHR0302) is a potent and orally active inhibitor of JAK family, particularly JAK1. Ivarmacitinib demonstrates more than 10-fold selectivity for JAK1 over JAK2, 77-fold over JAK3, and 420-fold over Tyk2. Ivarmacitinib also exhibits anti-proliferative and anti-inflammatory effects.
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