APS-2-79 HCl
Product Specifications
CAS Number
2002381-31-7
Target
MEK
Applications
Protein Tyrosine Kinase
Smiles
CC1=C (C=CC (=C1) OC2=CC=CC=C2) NC3=NC=NC4=CC (=C (C=C43) OC) OC.Cl
Molecular Formula
C23H21N3O3.HCl
Additionnal Information
APS-2-79 is a MAPK antagonist that modulating KSR-dependent MAPK signalling by antagonizing RAF heterodimerization as well as the conformational changes required for phosphorylation and activation of KSR-bound MEK. IC50=120 ± 23 nM.
Storage Conditions
2 years -80 in solvent
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
127898 100 µg
HLA-A (HLA Class I Histocompatibility Antigen, A-3 alpha Chain, MHC Class I Antigen A*3, HLAA)
Sign In for Pricing
View Details 
EK342667 96 Well
Rat PIIINP (N-Terminal Procollagen III Propeptide) ValidElisa Kit
Sign In for Pricing
View Details B7001 96 Tests
Astrocytic phosphoprotein PEA-15 (PEA15) Rat ELISA Kit
Sign In for Pricing
View Details