What is the catalog number for Antalarmin hydrochloride?

The catalog number for Antalarmin hydrochloride is E6536-5mg.

What sizes are available for Antalarmin hydrochloride?

Antalarmin hydrochloride is available in the following size(s): 5 mg.

Is Antalarmin hydrochloride in stock?

Antalarmin hydrochloride is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures Antalarmin hydrochloride?

Antalarmin hydrochloride is manufactured by Bimake.

What is the estimated delivery time for Antalarmin hydrochloride?

Estimated delivery time for Antalarmin hydrochloride is approximately 15 business day(s), depending on your location.

Antalarmin hydrochloride

Product Specifications

CAS Number

220953-69-5

Target

CRFR

Applications

GPCR & G Protein

Smiles

CC1=C (N2C (C) =C (C) C3=C (N (CCCC) CC) N=C (C) N=C32) C (C) =CC (C) =C1.[H]Cl

Molecular Formula

C24H35ClN4

Additionnal Information

Antalarmin hydrochloride is an orally active, non-peptide corticotropin-releasing hormone receptor 1 (CRHR1) antagonist exhibiting a Ki value of 1 nM. This compound inhibits CRH-induced ACTH secretion and attenuates CRH-mediated and novelty-induced anxiety-like behaviors in preclinical models. Additionally, antalarmin hydrochloride demonstrates anti-inflammatory activity in arthritis models and reduces stress-induced gastric ulceration associated with irritable bowel syndrome.