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GSK-843

Product Specifications

CAS Number

1601496-05-2

Synonyms

GSK'843

Target

RIP kinase

Applications

Apoptosis

Molecular Formula

C19H15N5S2

Additionnal Information

GSK-843 (GSK'843) is a selective inhibitor of receptor-interacting protein kinase 3 (RIP3 or RIPK3) that binds to the RIP3 kinase domain with an IC50 of 8.6 nM and effectively inhibits its enzymatic activity with an IC50 of 6.5 nM.
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