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TC14012

Product Specifications

CAS Number

368874-34-4

SKU

C04518-1mg

Additionnal Information

TC14012, a serum-stable derivative of T140, is a selective and peptidomimetic CXCR4 antagonist with an IC50 of 19.3 nM. TC14012 is a potent CXCR7 agonist with an EC50 of 350 nM for recruiting β-arrestin 2 to CXCR7. TC14012 has anti-HIV activity and anti-cancer activity.

Storage Conditions

3 years-20°C powder 2 years-80°C in solvent

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