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Suzetrigine

Product Specifications

CAS Number

2649467-58-1

Synonyms

VX-548

SKU

C01765-5mg

Target

Sodium Channel

Applications

Transmembrane Transporters

Additionnal Information

VX-548 (Suzetrigine), is an oral, highly selective inhibitor of voltage-gated sodium channel 1.8 (NaV1.8) with an IC50 of 0.7 nM. It can be used in research of transmitting nociceptive signals and treatment of acute pain after abdominoplasty or bunionectomy.

Available Sizes

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