CDK9 ligand-Linker Conjugate
CDK9 ligand-Linker Conjugate is a synthesized CDK9 ligand-linker conjugate that can be used for synthesis of dCDK9-202 (HY-178861) . dCDK9-202 is a potent CDK9 PROTAC degrader with anti-tumor activity[1].
Product Specifications
UNSPSC
12352005
Target
Target Protein Ligand-Linker Conjugates
Related Pathways
PROTAC
Field of Research
Cancer
Smiles
O=CCCCCCCCN1CC2=C(C1)C=C3C(N(C(C3=C2)=O)C4CCC(NC4=O)=O)=O
Molecular Formula
C23H27N3O5
Molecular Weight
425.48
References & Citations
[1]Ma L, et al. Discovery of dCDK9-202 as a Highly Potent and Selective PROTAC CDK9 Degrader with Strong In Vivo Antitumor Activity. J Med Chem. 2025 Oct 23;68 (20) :21172-21186.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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