LAS101057
LAS101057 is a potent, selective, and orally efficacious A2B receptor antagonist.
Product Specifications
CAS Number
925676-48-8
UNSPSC
12352005
Hazard Statement
H302, H315, H319, H335
Target
Adenosine Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Neuroscience-Neuromodulation
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/LAS101057.html
Purity
99.92
Solubility
DMSO : ≥ 125 mg/mL
Smiles
FC1=CN=CC=C1C(N=CC(NC(C2CC2)=O)=N3)=C3C4=CC=CN=C4
Molecular Formula
C18H14FN5O
Molecular Weight
335.34
Precautions
H302, H315, H319, H335
References & Citations
[1]Paul Eastwood, et al. Discovery of LAS101057: A Potent, Selective, and Orally Efficacious A2B Adenosine Receptor Antagonist. ACS Med Chem Lett. 2011 Mar 10; 2 (3) : 213-218.
Shipping Conditions
Room Temperature
Storage Conditions
4°C (Powder, protect from light)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
LC427793 20 µg
Invadolysin (LmLN) (NM_001136049) Human Over-expression Lysate
Sign In for Pricing
View Details 
