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GK718

Product Specifications

Target

HDAC

Related Pathways

DNA Damage/DNA Repair|||Chromatin/Epigenetic

Bioactivity

GK718, a selective HDAC1/3 inhibitor with IC50 values of 259 nM and 139 nM, respectively, elevates acetylated histone H3 levels in cells and mitigates Bleomycin-induced pulmonary fibrosis in mice [1].

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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