αO-Conotoxin GeXIVA
Product Specifications
CAS Number
2010167-25-4
Target
AChR
Related Pathways
Neuroscience
Bioactivity
αO-Conotoxin GeXIVA, a potent antagonist of the α9α10 nicotinic acetylcholine receptor (nAChR), exhibits an inhibition concentration 50 (IC50) of 12 nM against rat α9α10 nAChRs. This compound has demonstrated analgesic properties in animal pain models [1].
Molecular Formula
C139H227N55O41S4
Molecular Weight
3452.89
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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