Ep300/CREBBP-IN-8
Product Specifications
CAS Number
2259641-24-0
Target
Histone Acetyltransferase, Others
Related Pathways
Others, Chromatin/Epigenetic
Bioactivity
Ep300/CREBBP-IN-8 (Example 37), a potent and orally active inhibitor of Ep300 and CREBBP, shows IC50 values of 0.014 μM and 0.018 μM, respectively, and is utilized in cancer research [1].
Smiles
COc1ccc(cc1F)C1(CCCCC1)C(=O)N1C[C@H](F)C[C@@H]1C(=O)Nc1ccc2[nH]ncc2n1
Molecular Formula
C25H27F2N5O3
Molecular Weight
483.51
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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