Enzastaurin HCl
Product Specifications
CAS Number
359017-79-1
Target
Others, PKC, Autophagy, Apoptosis
Related Pathways
Others, Cytoskeletal Signaling, Chromatin/Epigenetic, Apoptosis, Autophagy
Bioactivity
Enzastaurin HCl, also known as DB-102 and LY317615, is a synthetic macrocyclic bisindolemaleimide with potential antineoplastic activity. Binding to the ATP-binding site, Enzastaurin HCl selectively inhibits protein kinase C beta, an enzyme involved in the induction of vascular endothelial growth factor (VEGF) -stimulated neo-angiogenesis. This agent may decrease tumor blood supply and so tumor burden.
Smiles
Cl.Cn1cc(C2=C(C(=O)NC2=O)c2cn(C3CCN(Cc4ccccn4)CC3)c3ccccc23)c2ccccc12
Molecular Formula
C32H30ClN5O2
Molecular Weight
552.08
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
Frequently Asked Questions
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