RS-102221
Product Specifications
CAS Number
185376-97-0
Target
5-HT Receptor
Related Pathways
GPCR/G Protein, Neuroscience
Bioactivity
RS-102221 is a selective antagonist of the 5-HT2C receptor with a K i of 10 nM, demonstrating nearly 100-fold more selectivity for the 5-HT2C receptor over the 5-HT2A and 5-HT2B receptors. This compound not only has the potential to promote the differentiation of new nerve cells but also increases food intake and weight gain in rats.
Smiles
O=C1NC(=O)C2(N1)CCN(CCCCC(=O)C3=CC(NS(=O)(=O)C4=CC=C(C=C4)C(F)(F)F)=C(OC)C=C3OC)CC2
Molecular Formula
C27H31F3N4O7S
Molecular Weight
612.62
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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