PKRA83 hydrochloride
Product Specifications
Target
Others
Related Pathways
Others
Bioactivity
PKRA83 (PKRA7) hydrochloride is a potent prokinetic (PK2) antagonist capable of crossing the blood-brain barrier, competitively inhibiting PK2 from binding to its receptors PKR1 and PKR2. It effectively suppresses PK2 receptors, with IC50 values of 5.0 nM for PKR1 and 8.2 nM for PKR2, and exhibits anticancer, anti-arthritis, and anti-angiogenic activities.
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
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