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PBRM1-BD2-IN-8

PBRM1-BD2-IN-8 (compound 34) is a potent PBRM1 Bromodomain inhibitor with PBRM1-BD2 Kd of 4.4 μM, PBRM1-BD2 IC50 of 0.16 μM, and PBRM1-BD5 Kd of 25 μM; PBRM1-BD2-IN-8 shows anti-cancer activity.

Product Specifications

CAS Number

2819989-75-6

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

317.18

Molecular Formula

C15H13BrN2O

Notes

Research use only, not for human use.

Receptor

Epigenetic Reader Domain

Available Sizes

Curated Selection

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