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LASSBio-1135

LASSBio-1135 is an orally effective antagonist of TRPV1 and inhibitor of TNF-α production.Oral administration of 100 mol x Kg (-1) LASSBio-1135 markedly reduced thermal hyperalgesia induced by carrageenan.

Product Specifications

CAS Number

852453-71-5

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

286.33

Molecular Formula

C18H14N4

Notes

Research use only, not for human use.

Receptor

TRPV1|TNF-α

Available Sizes

Curated Selection

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