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CU-CPT9b

CU-CPT9b is an antagonist of toll-like receptor 8 (TLR8; Kd = 21 nM) . It inhibits activation of NF-ĸB induced by the TLR8 agonist R-848 in TLR8-overexpressing HEK-Blue cells with an IC50 value of 0.7 nM.

Product Specifications

CAS Number

2162962-69-6

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

251.28

Molecular Formula

C16H13NO2

Notes

Research use only, not for human use.

Receptor

TLR8

Available Sizes

Curated Selection

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