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Pexmetinib

Pexmetinib (ARRY-614) is a potent, orally active, dual Tie-2/p38 MAPK inhibitor with IC50 of 1, 26 and 35 nM for Tie-2, p38α and p38β, respectively.

Product Specifications

CAS Number

945614-12-0

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

556.63

Molecular Formula

C31H33FN6O3

Notes

Research use only, not for human use.

Receptor

P38MAPK

Available Sizes

Curated Selection

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