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GSK1324726A

A potent and selective inhibitor of BET bromodomain with IC50 of 41 nM/31 nM/22 nM for BRD2/BRD3/BRD4 respectively.

Product Specifications

CAS Number

1300031-52-0

Stability

≥ 2 years

Purity

>98% (HPLC)

Weight

434.9147

Molecular Formula

C25H23ClN2O3

Notes

Research use only, not for human use.

Receptor

BRD2|BRD3|BRD4

Available Sizes

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