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ALKBH5-IN-5

ALKBH5-IN-5 is a potent and selective covalent inhibitor of the m6A demethylase ALKBH5 (IC50 = 0.62 μM) . It increases cellular m6A levels, demonstrating utility in vitro by promoting differentiation and apoptosis, supporting its investigation in oncology research, particularly in leukemia models.

Product Specifications

CAS Number

140481-05-6

Product Name Alternative

ALKBH5IN5

Field of Research

Cardiovascular Research, Metabolism Research, Signal Transduction

Purity

99.54% (May vary between batches)

Smiles

O=C1C=CC (=O) N1CCC=2C=CC=CC2OC

Molecular Formula

C13H13NO3

Molecular Weight

231.25

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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