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ENPP3 Inhibitor 1

ENPP3 Inhibitor 1 is a potent and selective small molecule targeting ENPP3 (IC50 = 0.15 μM), showing over 275-fold selectivity versus ENPP1. It has demonstrated antitumor activity in research models of breast and cervical cancer, supporting its use in oncology studies for investigating nucleotide signaling pathways in vitro and in vivo.

Product Specifications

CAS Number

2803505-90-8

Field of Research

Metabolism Research, Pharmacology & Drug Discovery

Smiles

O=C (NC1=CC=C (OS (=O) (=O) C2=CC=C (OC (F) (F) F) C=C2) C=C1) C=3C=CC=CC3

Molecular Formula

C20H14F3NO5S

Molecular Weight

437.39

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

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