EP1-antagonist-1
EP1-antagonist-1 is a potent and selective antagonist of the EP1 prostanoid receptor, exhibiting high affinity with a pKi of 7.54 and functional potency with a pIC50 of 8.5. This compound is a valuable research tool for investigating EP1 receptor function in models of pain, inflammation, and renal function in both in vitro and in vivo studies.
Product Specifications
CAS Number
851204-35-8
Product Name Alternative
Prostaglandin Receptor, ProstaglandinReceptor, EP1, EP1 antagonist 1, EP1-antagonist-1, EP1-antanoist-1
Field of Research
Immunology & Inflammation, Pharmacology & Drug Discovery
Purity
97.06% (May vary between batches)
Solubility
DMSO:55 mg/mL (116.99 mM)
Smiles
C (C1=C (OCC2=C (Cl) C=C (Cl) C=C2) C=CC (Br) =C1) N3N=C (C (O) =O) C=C3C
Molecular Formula
C19H15BrCl2N2O3
Molecular Weight
470.14
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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