CYT-1010
CYT-1010 is a potent and selective mu-opioid receptor agonist, demonstrating high functional bias with an EC50 of 0.0053 nM for inhibiting cAMP production versus 13.1 nM for β-arrestin recruitment. This profile makes it a valuable research tool for investigating biased agonism, G-protein signaling pathways, and pain-related in vitro and in vivo studies.
Product Specifications
CAS Number
213769-33-6
Field of Research
Metabolism Research, Neuroscience, Pharmacology & Drug Discovery
Smiles
C (C=1C=2C (NC1) =CC=CC2) [C@H]3C (=O) N[C@@H] (CC4=CC=CC=C4) C (=O) NCCCC[C@@H] (NC ([C@H] (CC5=CC=C (O) C=C5) N) =O) C (=O) N3
Molecular Formula
C35H40N6O5
Molecular Weight
624.73
Storage Conditions
-20°C
Notes
For research use only.
Available Sizes
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