CD161
CD161 is an orally active, selective BET bromodomain inhibitor with IC50 values of 28.2 nM and 7.2 nM for BRD4 BD1 and BD2, respectively. It demonstrates potent anticancer activity in cellular assays and has shown efficacy in in vivo tumor models, supporting its use in oncology and epigenetics research.
Product Specifications
CAS Number
1627716-22-6
Field of Research
Epigenetics & Chromatin, Immunology & Inflammation
Smiles
O (C) C=1C=C2C3=C (N=C (C) N=C3NC2=CC1C=4C (C) =NOC4C) C=5C6=C (N=CC5) C=CC=C6
Molecular Formula
C26H21N5O2
Molecular Weight
435.48
Storage Conditions
-20°C
Notes
For research use only.
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