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Aurora A/PKC-IN-1

Aurora A/PKC-IN-1 (Compound 2e) is a potent dual inhibitor of Aurora A and PKC isoforms, demonstrating low nanomolar IC50 values. It exhibits anti-proliferative and anti-metastatic activity in breast cancer cell studies, making it a valuable chemical probe for oncology research, particularly in studying kinase signaling pathways in vitro.

Product Specifications

CAS Number

2143100-98-3

Field of Research

Cell Biology, Epigenetics & Chromatin, Signal Transduction

Smiles

O=C1N ([Se]C=2C1=CC=CC2) C3=NC (NC4CC[Se]C4) =C5C (=N3) N=CN5

Molecular Formula

C16H14N6OSe2

Molecular Weight

464.24

Storage Conditions

-20°C

Notes

For research use only.

Available Sizes

Frequently Asked Questions

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