NPY5RA-972

NPY5RA-972 is an orally active, central nervous system (CNS) penetrating, potent and selective NPY Y5 receptor antagonist that prevents feeding driven by activation of this receptor[1].

Product Specifications

CAS Number

[439861-56-0]

UNSPSC

12352005

Hazard Statement

H302, H315, H319, H335

Target

Neuropeptide Y Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease

Assay Protocol

https://www.medchemexpress.com/npy5ra-972.html

Purity

98.99

Solubility

DMSO : 16.67 mg/mL (ultrasonic)

Smiles

O=C(N1CCOCC1)NC2=C(C)C(C3=CC=CC=C3N4C(C)C)=C4C=C2

Molecular Formula

C21H25N3O2

Molecular Weight

351.45

Precautions

H302, H315, H319, H335

References & Citations

[1]Andrew V Turnbull, et al. Selective antagonism of the NPY Y5 receptor does not have a major effect on feeding in rats. Diabetes. 2002 Aug;51 (8) :2441-9.