Derazantinib
Product Specifications
CAS Number
1234356-69-4
Target
FGFR
Related Pathways
Tyrosine Kinase/Adaptors, Angiogenesis
Purity
0.9995
Bioactivity
Derazantinib (ARQ-087) is a potent, ATP-competitive, orally active tyrosine kinase inhibitor with IC50 values of 4.5/1.8/4.35/3.4 nM for chondrocyte FGFR1/FGFR2/FGFR3/FGFR4, respectively.
Smiles
COCCNCCc1cccc(Nc2ncc3C[C@@H](c4ccccc4F)c4ccccc4-c3n2)c1
Molecular Formula
C29H29FN4O
Molecular Weight
468.57
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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