What is the catalog number for GSK778?

The catalog number for GSK778 is T9703.

What sizes are available for GSK778?

GSK778 is available in the following size(s): 1 mL - 10 mM (in DMSO), 1 mg, 5 mg, 10 mg, 25 mg, 50 mg, 100 mg.

How many pack sizes does GSK778 come in?

GSK778 is available in 7 different pack sizes.

GSK778 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures GSK778?

GSK778 is manufactured by Molfinity.

What is the estimated delivery time for GSK778?

Estimated delivery time for GSK778 is approximately 10 business day(s), depending on your location.

GSK778

Product Specifications

CAS Number

2451862-42-1

Target

Epigenetic Reader Domain, Apoptosis

Related Pathways

Apoptosis, Chromatin/Epigenetic

Purity

0.9842

Bioactivity

GSK778 is a potent and selective inhibitor of BD1 bromodomain such as BRD2 BD1 (IC50s = 75 nM), BRD3 BD1 (IC50s = 41 nM), BRD4 BD1 (IC50s = 41 nM), and BRDT BD1 (IC50s = 143 nM) . GSK778 inhibits proliferation, induces a cell cycle arrest and apoptosis.