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AMG319

Product Specifications

CAS Number

1608125-21-8

Target

PI3K

Related Pathways

PI3K/Akt/mTOR signaling

Purity

0.9924

Bioactivity

AMG319 is a potent and selective PI3K? inhibitor with an IC50 of 18 nM and exhibits >47-fold selectivity over other PI3Ks. [Phase 2]

Smiles

C[C@H](Nc1ncnc2[nH]cnc12)c1cc2ccc(F)cc2nc1-c1ccccn1

Molecular Formula

C21H16FN7

Molecular Weight

385.4

Shipping Conditions

Cool pack

Storage Temperature

-20°C

Available Sizes

Curated Selection

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