EPI-7170
Product Specifications
CAS Number
2139288-26-7
Target
Others, Androgen Receptor
Related Pathways
Others, Endocrinology/Hormones
Bioactivity
EPI-7170 is a ralaniten analogue and a potent antagonist of the androgen receptor N-terminal structural domain, blocking the transcriptional activity of the full-length AR (FL-AR) and AR splice variants (AR-Vs) . EPI-7170 exhibits antitumor activity against enzalutamide resistant debulking resistant prostate cancer (CRPC) .
Smiles
C(C)(C)(C1=CC(Cl)=C(OC[C@@H](CCl)O)C(Cl)=C1)C2=CC=C(OC[C@@H](CNS(C)(=O)=O)O)C=C2
Molecular Formula
C22H28Cl3NO6S
Molecular Weight
540.88
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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