CCG215022

1813527-81-9

PKA, GRK

GPCR/G Protein, Tyrosine Kinase/Adaptors

0.9969

CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM for GRK2, 0.38±0.06 μM for GRK5, and 3.9±1 μM for GRK1.

CC1=C(C(NC(=O)N1)c1ccc(F)c(c1)C(=O)NCc1ccccn1)C(=O)Nc1ccc2[nH]ncc2c1

C26H22FN7O3

499.5

Ice Packs

-20°C