PF-670462
Product Specifications
CAS Number
950912-80-8
Target
Casein Kinase
Related Pathways
Metabolism|||Stem Cells
Purity
0.9972
Bioactivity
PF-670462 is a potent (IC50 = 7.7 ± 2.2 nM) and selective (>30-fold with respect to 42 additional kinases) inhibitor of CK1? in isolated enzyme preparations.
Smiles
Cl.Cl.Nc1nccc(n1)-c1c(ncn1C1CCCCC1)-c1ccc(F)cc1
Molecular Formula
C19H22Cl2FN5
Molecular Weight
410.32
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
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