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CPI203

Product Specifications

CAS Number

202591-23-9

Target

Others, Epigenetic Reader Domain

Related Pathways

Others, Chromatin/Epigenetic

Purity

0.9977

Bioactivity

CPI203 (CPI 203) is an effective BET bromodomain inhibitor (IC50: 37 nM for BRD4) .

Smiles

CC=1C2=C(N3C(C(CC(N)=O)N=C2C4=CC=C(Cl)C=C4)=NN=C3C)SC1C

Molecular Formula

C19H18ClN5OS

Molecular Weight

399.9

Shipping Conditions

Ice Packs

Storage Temperature

-20°C

Available Sizes

Frequently Asked Questions

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