BI-3812
Product Specifications
CAS Number
2166387-64-8
Target
Bcl-2 Family|||Bcl-6
Related Pathways
Immunology/Inflammation|||Apoptosis
Purity
0.9979
Bioactivity
BI-3812 is an inhibitor of BCL6. Which inhibiting the BTB domain of BCL6 (IC50: 3 nM) . BI-3812 also has antitumor activity.
Smiles
CNC(=O)COc1cc2cc(Nc3nc(ncc3Cl)N3CCC(CC3)C(=O)N(C)C)cc(OC)c2n(C)c1=O
Molecular Formula
C26H32ClN7O5
Molecular Weight
558.03
Shipping Conditions
Cool pack
Storage Temperature
-20°C
Available Sizes
Curated Selection
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