GB-110
Product Specifications
CAS Number
1252806-70-4
Target
Others, Protease-activated Receptor
Related Pathways
Others, GPCR/G Protein
Bioactivity
GB-110 selectively induces PAR2-mediated intracellular Ca2+ release in HT29 cells with an EC50 of 0.28 μM. GB-110 is a potent, orally active, and nonpeptidic protease activated receptor 2 (PAR2) agonist.
Smiles
[C@H](CC1CCCCC1)(C(N[C@H](C(NCC2=CC(C(=O)N3CCC(CN)CC3)=CC=C2)=O)[C@H](CC)C)=O)NC(=O)C4=CC=NO4
Molecular Formula
C33H48N6O5
Molecular Weight
608.77
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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