CNX-500
Product Specifications
CAS Number
1202758-21-1
Target
Others, BTK
Related Pathways
Tyrosine Kinase/Adaptors, Angiogenesis, Others
Bioactivity
CNX-500, a probe comprising a covalent Btk inhibitor chemically linked to biotin, exhibits significant inhibitory activity against Btk (IC50: 0.5 nM) and can form a covalent bond with Btk. Additionally, CNX-500 has low inhibitory effects on kinase EGFR and upstream Src-family kinases.
Smiles
[H][C@]12CS[C@@H](CCCCC(=O)NCCCOCCOCCOCCCNC(=O)CCCC(=O)NCCCOc3cccc(Nc4ncc(C)c(Nc5cccc(NC(=O)C=C)c5)n4)c3)[C@@]1([H])NC(=O)N2
Molecular Formula
C48H68N10O9S
Molecular Weight
961.18
Shipping Conditions
Ice Packs
Storage Temperature
-20°C
Available Sizes
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