LPA5 antagonist 3

LPA5 antagonist 3 (Example 74) is a lysophosphatidic acid receptor 5 (LPA5) antagonist, with an IC50 of 170 nM. LPA5 antagonist 3 can be used for the research of pain disorders and atherosclerosis[1].

Product Specifications

CAS Number

[1664336-44-0]

UNSPSC

12352005

Target

LPL Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease; Cardiovascular Disease

Assay Protocol

https://www.medchemexpress.com/lpa5-antagonist-3.html

Solubility

10 mM in DMSO

Smiles

O=C(C1=CC=C(CN(CC(F)(C)F)C(C2=CC=C(C=C2)OC3=C(F)C=CC=C3)=O)C=C1)O

Molecular Formula

C24H20F3NO4

Molecular Weight

443.42

References & Citations

[1]BUFFHAM W, et al. Amide derivatives as lysophosphatidic acid receptor antagonists. WO2015025164A1. 2015-02-26.

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Curated Selection

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